Synthesis of Indoles through Palladium-Catalyzed Three-Component Reaction of Aryl Iodides, Alkynes, and Diaziridinone

array(2) { ["lab"]=> string(3) "361" ["publication"]=> string(4) "4730" } Synthesis of Indoles through Palladium-Catalyzed Three-Component Reaction of Aryl Iodides, Alkynes, and Diaziridinone - 张扬会课题组 | LabXing

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2018

期刊 Organic Letters

作者 Bo Zhou · Zhuo Wu · Ding Ma · Xiaoming Ji · Yanghui Zhang

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The three-component reaction of aryl iodides, alkynes, and diaziridinone is described. The reaction provides an innovative synthetic approach for indoles. The approach features high efficiency, broad substrate scope, and excellent regioselectivity. C,C-Palladacycles should act as the intermediates. The C,C-palladacycles are obtained from simple aryl halides and alkynes and then reacted with diaziridinone to afford indoles.

卷 20
期 20
页码 6440-6443
American Chemical Society (ACS)
ISSN: 1523-7060
DOI: 10.1021/acs.orglett.8b02750

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